Addition of E138K to R263K in HIV integrase increases resistance to dolutegravir, but fails to restore activity of the HIV integrase enzyme and viral replication capacity

Thibault Mesplède, Nathan Osman, Melissa Wares, Peter K. Quashie, Said Hassounah, Kaitlin Anstett, Yingshan Han, Diane N. Singhroy, Mark A. Wainberg

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Pharmacology, Toxicology and Pharmaceutical Science

Immunology and Microbiology